Aromatase Inhibitors on steroid cyclesThis is the reason as to why Primobolan is often pitted against and compared to its close brother, Anavar. This is, does primobolan block estrogen, where the similarities between the two end, as Primobolan is an anabolic steroid that does primobolan block estrogen not only a weak affinity for various side effects, but also a weak anabolic strength when compared to the majority of other anabolic steroids in existence and in comparison to Anavar. Primobolan is a DHT-derivative anabolic steroid, which means it does not exhibit any interaction with the aromatase enzyme at any dose and therefore Primobolan does primobolan block estrogen effects olimp anabolic amino 5500 einnahme completely void of any Estrogenic side effects. Estrogen -related side effects such as water retention, rising blood pressure as a result of water retention and gynecomastia are nonexistent from Primobolan alone. Although Primobolan possesses a very low androgenic strength rating in comparison to Testosterone, Primobolan might still exhibit androgenic side effects especially in individuals with a greater sensitivity to this category of Primobolan side effects.
PRIMOBOLAN (Methenolone Enanthate) | omosironews.info
Many readers of this book will have already used steroids in the past, or are currently on a cycle to reach one goal or another. In the following text I will go a little more in-depth than just cursory knowledge and hopefully not bore to death those that already have some comprehension of the basic facts.
Successful dieting can also be sabotaged by the presence of high estrogen levels and lead to possible development of female fat pattern distribution in males, i. In women, progesterone will up to a certain point increase sex drive and then have the opposite effect when blood concentrations get too high. Even with a reduction of estrogens, they can still cause gynaecomastia in some users due to their overt activity at the progesterone receptor itself see Chapter 10 for more information on these specific compounds.
Which steroids do aromatise? Seen under the names: Foil strips of 10 tablets any dose , strips per box; bottles of 20, 30, 50 or tablets.
Developing swollen mammary glands in males is in the majority of cases non-life threatening, but that swollen gland can attract stubborn fat in the long-term, and might need surgical removal at a later date to rid the user of the unsightly lumps. Many users of tamoxifen think that it will help reduce water retention caused by the use of aromatising steroids, but this thought is flawed. So it will not prevent water retention in the aromatising steroid user or lower blood pressure from the higher plasma content in the blood caused by the rise in estrogens.
It has some other positive effects as well, and not just as a treatment of steroidal side effects. See more on this in the upcoming section on post cycle therapy. Another positive for tamoxifen is that it acts like some other triphenylethylene compounds by acting as an estrogen in the liver cells.
Rather than use the anti-aromatases to manage the estrogens, tamoxifen may be a better bet to keep the liver functioning normally, or even a low dose combination of both blockers and anti-aromatases to get the best of both worlds; slightly lower overall estrogen from the aromatase inhibitors AND some liver cell boosting effects to improve cholesterol from the tamoxifen. Tamoxifen was first synthesised in by chemical giant ICI.
Initially used as a treatment for certain forms of female infertility, it became available on the commercial market in the U. In , clinical trials of the drug began investigating its possible use as a combatant against breast cancer.
Amazingly, even with all the proven successes with tamoxifen, AstraZeneca discontinued the sale of Nolvadex in the U. In bodybuilding, a preventative dose for gynaecomastia in men is mg per day.
If a chap is not taking tamoxifen and develops swelling of the mammary gland, I suggest an immediate ingestion of 50mg or so to get the dose of tamoxifen up in the blood, then drop to mg for the rest of the cycle, or as long as the swelling persists. Much anecdotal evidence has suggested that this compound can influence a marked reduction in GH and IGF-1 production in the body; two VERY important hormones that AAS users attempt to maintain or even increase to promote synergistic growth.
Many athletes report minimised gains on light to moderate dosage AAS cycles when tamoxifen is used as an adjunct compared to when it is omitted entirely. Scientists have a theory that estrogens are actually needed in the body to keep the androgen receptors open discussed elsewhere , making for larger gains in mass and strength. For these negative reasons, users must weigh up whether the estrogenic side effect of gynaecomastia or negative blood lipid balance are enough of a problem to warrant tamoxifen use, particularly in the lighter androgenic cycles where gains might become negligible.
Many users actually wait until side effects become too problematic and then hit the tamoxifen at a relatively high dosage for one week as mentioned above , then taper down to just mg per day for the remnants of their cycle, which should not limit the big gains too much and is also more economically viable.
Please remember that I am talking with experience when I say that once gynaecomastia has started to develop it is almost impossible to regress its growth once initiated; the user must think very carefully before playing this hormonal form of Russian Roulette but the letrozole is always there as a back-up…see later.
Stopping the use of tamoxifen abruptly at any point when estrogen levels are at higher than normal levels, can cause a severe rebound of side effects which will onset rapidly. If a user is taking tamoxifen as an adjunct when on a steroid cycle it is best to stop its use when estrogen levels are at a more acceptable range, i.
Some other listed adverse effects are skin rashes, reduced white blood cell count and concurrent drop in immune system, visual disturbances, uterine fibroids and womb lining thickness changes, deep vein thrombosis leading to pulmonary embolism DVT , changes in liver enzymes and changes in blood lipids. To top things off, some women using tamoxifen have had an increased incidence of endometrial cancer and uterine sarcoma, as well as possible birth defects in the unknowingly pregnant.
So, a lady should think long and hard before adding tamoxifen into the mix just to get a little leaner or a little faster, especially when taking other drugs definitely not intended for use in the female metabolism. Frontloading with mg if gynaecomastia is being initially treated. No more than 10 mg daily for short period just prior to competition. Please note that this excerpt is only a small sample of the book chapter it is taken from. A great deal more content is available on this and many other topics in the Break the Code book.
The War on Female Hormones. Tamoxifen Citrate Seen under the names: Order your copy of Break The Code today! Excerpts from Break The Code.